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Molecular Characterization of c-Abl/c-Src Kinase Inhibitors Targeted against Murine Tumour Progenitor Cells that Express Stem Cell Markers

BACKGROUND: The non-receptor tyrosine kinases c-Abl and c-Src are overexpressed in various solid human tumours. Inhibition of their hyperactivity represents a molecular rationale in the combat of cancerous diseases. Here we examined the effects of a new family of pyrazolo [3,4-d] pyrimidines on a pa...

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Библиографические подробности
Главные авторы: Kruewel, Thomas, Schenone, Silvia, Radi, Marco, Maga, Giovanni, Rohrbeck, Astrid, Botta, Maurizio, Borlak, Juergen
Формат: Artigo
Язык:Inglês
Опубликовано: Public Library of Science 2010
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2994747/
https://ncbi.nlm.nih.gov/pubmed/21152443
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0014143
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