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Ethidium derivatives bind to G-quartets, inhibit telomerase and act as fluorescent probes for quadruplexes

The telomeric G-rich single-stranded DNA can adopt in vitro an intramolecular quadruplex structure, which has been shown to directly inhibit telomerase activity. The reactivation of this enzyme in immortalized and most cancer cells suggests that telomerase is a relevant target in oncology, and telom...

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Detaylı Bibliyografya
Asıl Yazarlar: Koeppel, Florence, Riou, Jean-François, Laoui, Abdelazize, Mailliet, Patrick, Arimondo, Paola B., Labit, Delphine, Petitgenet, Odile, Hélène, Claude, Mergny, Jean-Louis
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Oxford University Press 2001
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC29720/
https://ncbi.nlm.nih.gov/pubmed/11222758
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