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Chemistry and Pharmacological Characterization of Novel Nitrogen Analogs of AMOP-H-OH (Sazetidine-A; 6-[5-(Azetidin-2-ylmethoxy)pyridin-3-yl]hex-5-yn-1-ol) as α4β2-Nicotinic Acetylcholine Receptor-Selective Partial Agonists

In order to advance therapeutic applications of nicotinic ligands, continuing research efforts are being directed toward the identification and characterization of novel nicotinic acetylcholine receptor (nAChR) ligands that are both potent and subtype selective. Herein we report the synthesis and ph...

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Autori principali: Liu, Jianhua, Eaton, J. Brek, Caldarone, Barbara, Lukas, Ronald J., Kozikowski, Alan P.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2957884/
https://ncbi.nlm.nih.gov/pubmed/20822184
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm100765u
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