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Targeting SDF-1/CXCL12 with a ligand that prevents activation of CXCR4 through structure based drug design

[Image: see text] CXCL12 is an attractive target for clinical therapy because of its involvement in autoimmune diseases, cancer growth, metastasis, and neovascularization. Tyrosine sulfation at three positions in the CXCR4 N-terminus is crucial for specific, high-affinity CXCL12 binding. An NMR stru...

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Autors principals: Veldkamp, Christopher T., Ziarek, Joshua J., Peterson, Francis C., Chen, Yu, Volkman, Brian F.
Format: Artigo
Idioma:Inglês
Publicat: 2010
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2941798/
https://ncbi.nlm.nih.gov/pubmed/20459090
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja1002263
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