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Photo-cytotoxic trans diam(m)ine platinum(IV) diazido complexes more potent than their cis isomers

The photocytotoxicity of a series of anticancer trans-dihydroxido [Pt(N(3))(2)(OH)(2)(NH(3))(X)] (X = alkyl or aryl amine) platinum(IV) diazido complexes has been examined and the influence of cis-trans isomerism investigated. A series of photoactivatable Pt(IV)-azido complexes has been synthesized:...

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Detalhes bibliográficos
Main Authors: Farrer, Nicola J., Woods, Julie A., Munk, Vivienne P., Mackay, F. S., Sadler, Peter J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2933822/
https://ncbi.nlm.nih.gov/pubmed/19994893
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/tx900372p
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