Caricamento...

Structure-based design, synthesis, and biological evaluation of lipophilic-tailed monocationic inhibitors of neuronal nitric oxide synthase

Selective inhibitors of neuronal nitric oxide synthase (nNOS) have the potential to develop into new neurodegenerative therapeutics. Recently, we described the discovery of novel nNOS inhibitors (1a and 1b) based on a cis-pyrrolidine pharmacophore. These compounds and related ones were found to have...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Xue, Fengtian, Huang, Jinwen, Ji, Haitao, Fang, Jianguo, Li, Huiying, Martásek, Pavel, Roman, Linda J., Poulos, Thomas L., Silverman, Richard B.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2925225/
https://ncbi.nlm.nih.gov/pubmed/20673724
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2010.06.074
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !