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Histone Deacetylase Inhibitor MS-275 Exhibits Poor Brain Penetration: Pharmacokinetic Studies of [(11)C]MS-275 using Positron Emission Tomography

[Image: see text] MS-275 (entinostat) is a histone deacetylase (HDAC) inhibitor currently in clinical trials for the treatment of several types of cancer. Recent reports have noted that MS-275 can cross the blood−brain barrier (BBB) and cause region-specific changes in rodent brain histone acetylati...

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Detaylı Bibliyografya
Asıl Yazarlar: Hooker, Jacob M., Kim, Sung Won, Alexoff, David, Xu, Youwen, Shea, Colleen, Reid, Alicia, Volkow, Nora, Fowler, Joanna S.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Chemical Society 2009
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC2908422/
https://ncbi.nlm.nih.gov/pubmed/20657706
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cn9000268
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