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Proton pump inhibitor Lansoprazole is a nuclear Liver X Receptor agonist

The liver X receptors (LXRα and LXRβ) are transcription factors that control the expression of genes primarily involved in cholesterol metabolism. In brain, in addition to normal neuronal function, cholesterol metabolism is important for APP proteolytic cleavage, secretase activities, Aβ aggregation...

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Detalhes bibliográficos
Main Authors: Cronican, Andrea A., Fitz, Nicholas F., Pham, Tam, Fogg, Allison, Kifer, Brionna, Koldamova, Radosveta, Lefterov, Iliya
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2834822/
https://ncbi.nlm.nih.gov/pubmed/20060385
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2009.12.018
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