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Proton pump inhibitor Lansoprazole is a nuclear Liver X Receptor agonist

The liver X receptors (LXRα and LXRβ) are transcription factors that control the expression of genes primarily involved in cholesterol metabolism. In brain, in addition to normal neuronal function, cholesterol metabolism is important for APP proteolytic cleavage, secretase activities, Aβ aggregation...

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Dettagli Bibliografici
Autori principali: Cronican, Andrea A., Fitz, Nicholas F., Pham, Tam, Fogg, Allison, Kifer, Brionna, Koldamova, Radosveta, Lefterov, Iliya
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2834822/
https://ncbi.nlm.nih.gov/pubmed/20060385
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2009.12.018
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