Carregant...

Synthesis and In Vitro Evaluation of Aspartate Transcarbamoylase Inhibitors

The design, synthesis, and evaluation of a series of novel inhibitors of aspartate transcarbamoylase (ATCase) are reported. Several submicromolar phosphorus-containing inhibitors are described, but all-carboxylate compounds are inactive. Compounds were synthesized to probe the postulated cyclic tran...

Descripció completa

Guardat en:
Dades bibliogràfiques
Autors principals: Coudray, Laëtitia, Pennebaker, Anne F., Montchamp, Jean-Luc
Format: Artigo
Idioma:Inglês
Publicat: 2009
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2783949/
https://ncbi.nlm.nih.gov/pubmed/19828320
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2009.09.045
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!