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Discriminative Stimulus Effects of 1-(2,5-Dimethoxy-4-methylphenyl)-2-aminopropane (DOM), Ketanserin, and (R)-(+)-α-(2,3-Dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in Rats

Very little is known about constitutive activity in vivo. This study examined whether constitutive activity and inverse agonism contribute to discriminative stimulus effects of drugs acting at serotonin (5-HT)(2A) receptors. Rats were trained to discriminate between saline and either 0.56 mg/kg 5-HT...

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Autori principali: Li, Jun-Xu, Unzeitig, Alison, Javors, Martin A., Rice, Kenner C., Koek, Wouter, France, Charles P.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2775261/
https://ncbi.nlm.nih.gov/pubmed/19687292
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.109.157560
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