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Novel topoisomerase I-targeting antitumor agents synthesized from the N,N,N-trimethylammonium derivative of ARC-111, 5H-2,3-dimethoxy-8,9-methylenedioxy-5-[(2-N,N,N-trimethylammonium)ethyl]dibenzo[c,h][1,6]-naphthyridin-6-one iodide

Several new TOP1-targeting agents were prepared using as an intermediate the N,N,N-trimethyl quaternary ammonium salt 2 of ARC-111. Direct displacement of the quaternary ammonium group with hydroxide, cyclopropylamine, imidazole, 1H-1,2,3-triazole, alkylethylenediamines, ethanolamine, and polyhydrox...

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Hlavní autoři: Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2009
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2766012/
https://ncbi.nlm.nih.gov/pubmed/19299037
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2009.02.004
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