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Acute dasatinib exposure commits Bcr-Abl–dependent cells to apoptosis

Pioneering work with the Bcr-Abl inhibitor, imatinib, demonstrated a requirement for constant Bcr-Abl inhibition to achieve maximal therapeutic benefit in treating chronic myeloid leukemia (CML), establishing a paradigm that has guided further drug development for this disease. Surprisingly, the sec...

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Dades bibliogràfiques
Autors principals: Snead, Jennifer L., O'Hare, Thomas, Adrian, Lauren T., Eide, Christopher A., Lange, Thoralf, Druker, Brian J., Deininger, Michael W.
Format: Artigo
Idioma:Inglês
Publicat: American Society of Hematology 2009
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2765681/
https://ncbi.nlm.nih.gov/pubmed/19706883
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2007-10-113969
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