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Synthesis and In Vivo Antitumor Efficacy of PEGylated Poly(L-lysine) Dendrimer-Camptothecin Conjugates

Polymer conjugates of camptothecin (CPT) have been pursued as a solution to the difficulties present in treating cancers with CPT and its derivatives. Covalent attachment of CPT to a polymer can improve solubility, increase blood circulation time, enhance tumor uptake, and significantly improve effi...

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Autori principali: Fox, Megan E., Guillaudeu, Steve, Fréchet, Jean M. J., Jerger, Kat, Macaraeg, Nichole, Szoka, Francis C.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2765109/
https://ncbi.nlm.nih.gov/pubmed/19588994
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/mp9001206
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