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Antineoplastic Agents 552. Oxidation of Combretastatin A-1: Trapping the o-Quinone Intermediate Considered the Metabolic Product of the Corresponding Phosphate Prodrug 1

The very unstable (< 10 min at rt) o-quinone (5) derived from the vicinal diphenol anticancer drug combretastatin A-1 (1) has been obtained by careful oxidation with NaIO(4) and tetrabutylammonium bromide in water/dichloromethane. Immediate reaction with phenylenediamine (6) allowed o-quinone 5 t...

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Detalhes bibliográficos
Main Authors: Pettit, George R., Thornhill, Andrew J., Moser, Bryan R., Hogan, Fiona
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2756244/
https://ncbi.nlm.nih.gov/pubmed/18729517
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/np800179g
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