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Design, Synthesis, Biological Evaluation, and Structural Characterization of Potent Histone Deacetylase Inhibitors Based on Cyclic α/β-Tetrapeptide Architectures

Histone deacetylases (HDACs) are a family of enzymes found in bacteria, fungi, plants, and animals that profoundly affect cellular function by catalyzing the removal of acetyl groups from ε-N-acetylated lysine residues of various protein substrates including histones, transcription factors, α-tubuli...

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Autores principales: Montero, Ana, Beierle, John M., Olsen, Christian A., Ghadiri, M. Reza
Formato: Artigo
Lenguaje:Inglês
Publicado: 2009
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2751792/
https://ncbi.nlm.nih.gov/pubmed/19239270
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja809508f
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