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No increase in breast cancer recurrence with concurrent use of tamoxifen and some CYP2D6-inhibiting medications

Tamoxifen reduces recurrence risk among women treated for estrogen receptor-positive breast cancer. Its effectiveness partly depends on metabolic activation via cytochrome P450 2D6 (CYP2D6). Some medications compromise CYP2D6 activity and may lower plasma concentrations of active tamoxifen metabolit...

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Detalhes bibliográficos
Main Authors: Ahern, Thomas P., Pedersen, Lars, Cronin-Fenton, Deirdre P., Sørensen, Henrik Toft, Lash, Timothy L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2742564/
https://ncbi.nlm.nih.gov/pubmed/19690182
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1055-9965.EPI-09-0516
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