Loading...

An all-atom model for stabilization of α-helical structure in peptides by hydrocarbon staples

Recent work has shown that the incorporation of an all-hydrocarbon “staple” into peptides can greatly increase their α-helix propensity, leading to an improvement in pharmaceutical properties such as proteolytic stability, receptor affinity and cell-permeability. Stapled peptides thus show promise a...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Main Authors: Kutchukian, Peter S., Yang, Jae Shick, Verdine, Gregory L., Shakhnovich, Eugene I.
Format: Artigo
Sprog:Inglês
Udgivet: 2009
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2735086/
https://ncbi.nlm.nih.gov/pubmed/19334772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja805037p
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!