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Modeling the Autoinhibition of Clarithromycin Metabolism during Repeated Oral Administration

Clarithromycin decreases CYP3A4 activity and thus gradually inhibits its own metabolism as well as that of coadministered drugs. The aim of this study was to obtain an understanding of the time course of these changes. The plasma concentration-time profiles of clarithromycin and its active metabolit...

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Autori principali: Abduljalil, Khaled, Kinzig, Martina, Bulitta, Jürgen, Horkovics-Kovats, Stefan, Sörgel, Fritz, Rodamer, Michael, Fuhr, Uwe
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology (ASM) 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2704653/
https://ncbi.nlm.nih.gov/pubmed/19414584
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01193-08
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