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Path integral method for predicting relative binding affinities of protein-ligand complexes

We present a novel approach for computing biomolecular interaction binding affinities based on a simple path integral solution of the Fokker-Planck equation. Computing the free energy of protein-ligand interactions can expedite structure-based drug design. Traditionally, the problem is seen through...

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Autori principali: Mulakala, Chandrika, Kaznessis, Yiannis N.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2671935/
https://ncbi.nlm.nih.gov/pubmed/19275144
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja807460s
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