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Membrane Hyperpolarization Drives Cation Influx and Fungicidal Activity of Amiodarone

Cationic amphipathic drugs, such as amiodarone, interact preferentially with lipid membranes to exert their biological effect. In the yeast Saccharomyces cerevisiae, toxic levels of amiodarone trigger a rapid influx of Ca(2+) that can overwhelm cellular homeostasis and lead to cell death. To better...

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Autori principali: Maresova, Lydie, Muend, Sabina, Zhang, Yong-Qiang, Sychrova, Hana, Rao, Rajini
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2631971/
https://ncbi.nlm.nih.gov/pubmed/19054772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M806693200
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