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Discovery of 1,4-Didydroxy-2-naphthoate Prenyltransferase Inhibitors: New Drug Leads for Multidrug-Resistant Gram-Positive Pathogens

Since utilization of menaquinone in the electron transport system is a characteristic of Gram-positive organisms, the 1,4-dihydroxy-2-naphthoate prenyltransferase (MenA) inhibitors 1a and 2a act as selective antibacterial agents against organisms such as methicillin-resistant Stapylococcus aureus (M...

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Detalhes bibliográficos
Main Authors: Kurosu, Michio, Narayanasamy, Prabagaran, Biswas, Kallolmay, Dhiman, Rakesh, Crick, Dean C.
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2591091/
https://ncbi.nlm.nih.gov/pubmed/17658779
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm070638m
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