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In Vitro Plasma Stability, Permeability and Solubility of Mercaptoacetamide Histone Deacetylase Inhibitors

Histone deacetylase inhibitors (HDACIs) are emerging as a new class of therapeutic agents with potent antitumor activities in a broad spectrum of human cancers. In this study, the in vitro plasma stability, permeability, solubility, and lipophilicity (logD) of two mercaptoacetamide-based HDACIs (cod...

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Библиографические подробности
Главные авторы: Konsoula, Roula, Jung, Mira
Формат: Artigo
Язык:Inglês
Опубликовано: 2008
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2565275/
https://ncbi.nlm.nih.gov/pubmed/18562136
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijpharm.2008.05.001
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