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Synthesis of (±)-Brazilin Using IBX

A short synthesis of (±)-brazilin is reported. This synthesis uses several interesting and underutilized transformations including a regioselective dirhodium-catalyzed aryl C–H insertion, a regioselective IBX phenol → o-quinone oxidation, a tautomerization of an o-quinone to a p-quinone methide, and...

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Autors principals: Huang, Yaodong, Zhang, Jinsong, Pettus, Thomas R. R.
Format: Artigo
Idioma:Inglês
Publicat: 2005
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2423948/
https://ncbi.nlm.nih.gov/pubmed/16354080
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/o1023749
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