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Rational Design and Generation of a Bimodal Bifunctional Ligand for Antibody-Targeted Radiation Cancer Therapy

An antibody-targeted radiation therapy (radioimmunotherapy, RIT) employs a bifunctional ligand that can effectively hold a cytotoxic metal with clinically acceptable complexation kinetics and stability while being attached to a tumor-specific antibody. Clinical exploration of the therapeutic potenti...

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Autors principals: Chong, Hyun-Soon, Ma, Xiang, Le, Thien, Kwamena, Baidoo, Milenic, Diane E., Brady, Erik D., Song, Hyun A., Brechbiel, Martin W.
Format: Artigo
Idioma:Inglês
Publicat: 2007
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2396554/
https://ncbi.nlm.nih.gov/pubmed/18062661
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm070401q
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