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Deltorphin transport across the blood–brain barrier

In vivo antinociception studies demonstrate that deltorphins are opioid peptides with an unusually high blood–brain barrier penetration rate. In vitro, isolated bovine brain microvessels can take up deltorphins through a saturable nonconcentrative permeation system, which is apparently distinct from...

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Bibliografiske detaljer
Udgivet i:Proc Natl Acad Sci U S A
Principais autores: Fiori, Anna, Cardelli, Patrizia, Negri, Lucia, Savi, Maria Rosaria, Strom, Roberto, Erspamer, Vittorio
Format: Artigo
Sprog:Inglês
Udgivet: National Academy of Sciences 1997
Fag:
Online adgang:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC23226/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/9256506/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.94.17.9469
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