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Deltorphin transport across the blood–brain barrier

In vivo antinociception studies demonstrate that deltorphins are opioid peptides with an unusually high blood–brain barrier penetration rate. In vitro, isolated bovine brain microvessels can take up deltorphins through a saturable nonconcentrative permeation system, which is apparently distinct from...

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Dades bibliogràfiques
Publicat a:Proc Natl Acad Sci U S A
Autors principals: Fiori, Anna, Cardelli, Patrizia, Negri, Lucia, Savi, Maria Rosaria, Strom, Roberto, Erspamer, Vittorio
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 1997
Matèries:
Accés en línia:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC23226/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/9256506/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.94.17.9469
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