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Improved Oral Bioavailability and Brain Transport of Saquinavir Upon Administration in Novel Nanoemulsion Formulations

The aim of this investigation was to develop novel oil-in-water (o/w) nanoemulsions containing saquinavir (SQV), an anti-HIV protease inhibitor, for enhanced oral bioavailability and brain disposition. SQV was dissolved in different types of edible oils rich in essential polyunsaturated fatty acids...

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Autori principali: Vyas, Tushar K., Shahiwala, Aliasgar, Amiji, Mansoor M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2007
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2213794/
https://ncbi.nlm.nih.gov/pubmed/17651927
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijpharm.2007.06.016
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