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Contribution of the active metabolite M1 to the pharmacological activity of tesofensine in vivo: a pharmacokinetic-pharmacodynamic modelling approach

BACKGROUND AND PURPOSE: Tesofensine is a centrally acting drug under clinical development for Alzheimer's disease, Parkinson's disease and obesity. In vitro, the major metabolite of tesofensine (M1) displayed a slightly higher activity, which however has not been determined in vivo. The ai...

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Autori principali: Lehr, T, Staab, A, Tillmann, C, Nielsen, E Ø, Trommeshauser, D, Schaefer, H G, Kloft, C
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2007
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2199391/
https://ncbi.nlm.nih.gov/pubmed/17982477
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0707539
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