Aminophosphinic inhibitors as transition state analogues of enkephalin-degrading enzymes: A class of central analgesics

Lignende værker

• Structure of aminopeptidase N from Escherichia coli complexed with the transition‐state analogue aminophosphinic inhibitor PL250
  af: Fournié‐Zaluski, Marie‐Claude, et al.
  Udgivet: (2009)
• Long-lasting oral analgesic effects of N-protected aminophosphinic dual ENKephalinase inhibitors (DENKIs) in peripherally controlled pain
  af: Bonnard, Elisabeth, et al.
  Udgivet: (2015)
• Enhancement of the effects of a complete inhibitor of enkephalin-catabolizing enzymes, RB 101, by a cholecystokinin-B receptor antagonist in diabetic rats
  af: Coudoré-Civiale, Marie-Ange, et al.
  Udgivet: (2001)
• Design of the first highly potent and selective aminopeptidase N (EC 3.4.11.2) inhibitor
  af: Huixiong Chen, et al.
  Udgivet: (1999)
• Similar decrease in spontaneous morphine abstinence by methadone and RB 101, an inhibitor of enkephalin catabolism.
  af: Ruiz, F., et al.
  Udgivet: (1996)