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Substrate- and pH-dependent contribution of oxyanion binding site to the catalysis of prolyl oligopeptidase, a paradigm of the serine oligopeptidase family.

Prolyl oligopeptidase, an enzyme implicated in memory disorders, is a member of a new serine peptidase family. Crystallographic studies (Fülöp et al., 1998) revealed a novel oxyanion binding site containing a tyrosine residue, Tyr473. To study the importance of Tyr473 OH, we have produced prolyl oli...

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Библиографические подробности
Главные авторы: Szeltner, Z., Renner, V., Polgár, L.
Формат: Artigo
Язык:Inglês
Опубликовано: Cold Spring Harbor Laboratory Press 2000
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2144544/
https://ncbi.nlm.nih.gov/pubmed/10716187
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