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Predicting absolute ligand binding free energies to a simple model site

A central challenge in structure-based ligand design is the accurate prediction of binding free energies. Here, we apply alchemical free energy calculations in explicit solvent to predict ligand binding in a model cavity in T4 lysozyme. Even in this simple site, there are challenges. We made systema...

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Bibliografske podrobnosti
Main Authors: Mobley, David L., Graves, Alan P., Chodera, John D., McReynolds, Andrea C., Shoichet, Brian K., Dill, Ken A.
Format: Artigo
Jezik:Inglês
Izdano: 2007
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2104542/
https://ncbi.nlm.nih.gov/pubmed/17599350
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jmb.2007.06.002
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