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Differential inhibition of cytochrome P450 isoforms by the protease inhibitors, ritonavir, saquinavir and indinavir

Aims To compare the inhibitory potential of the HIV protease inhibitors saquinavir, ritonavir and indinavir against CYP1A2, CYP2C9, CYP2E1 and CYP3A4 catalysed metabolic reactions in human liver microsomes in vitro. Methods Microsomes from six human livers were utilized in this study. The probe subs...

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Main Authors: Eagling, V. A., Back, D. J., Barry, M. G.
Formato: Artigo
Idioma:Inglês
Publicado: 1997
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2042821/
https://ncbi.nlm.nih.gov/pubmed/9278209
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1046/j.1365-2125.1997.00644.x
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