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Synthesis of (6R)- and (6S)-5,10-dideazatetrahydrofolate oligo-γ-glutamates: Kinetics of multiple glutamate ligations catalyzed by folylpoly-γ-glutamate synthetase

Folylpoly-γ-glutamate synthetase (FPGS, EC 6.3.2.17) catalyzes the ATP-dependent ligation of glutamic acid to reduced folates including (6S)-5,6,7,8-tetrahydrofolate (H(4)PteGlu), as well as to anticancer drugs such as 5,10-dideaza-5,6,7,8-tetrahydrofolate ((6R)-DDAH(4)PteGlu(1), (6R)-DDATHF, Lometr...

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Hlavní autoři: Tomsho, John W., McGuire, John J., Coward, James K.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2005
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1989673/
https://ncbi.nlm.nih.gov/pubmed/16132101
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/b505907k
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