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Pro- and anti-convulsant properties of PK 11195, a ligand for benzodiazepine binding sites: development of tolerance.

Ro 5-4864 is a benzodiazepine that differs from diazepam only in a p-chloro substituent and yet is inactive at the classical CNS binding sites. However it is a potent ligand for the peripheral type of benzodiazepine binding sites. PK 11195 is an isoquinoline carboxamide derivative that potently disp...

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Библиографические подробности
Главный автор: File, S. E.
Формат: Artigo
Язык:Inglês
Опубликовано: Nature Publishing Group 1984
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC1987107/
https://ncbi.nlm.nih.gov/pubmed/6091832
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