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Is Ro 03-7894 an irreversible antagonist at beta-adrenoceptor sites?

Ro 03-7894 (0.6 mM) produced a non-parallel shift to the right of dose-response curves to (-)-isoprenaline in K+ depolarized uterine preparations from the guinea-pig. The displacement of the curves was readily reversed by washing. A rightward shift of similar magnitude was also produced by Ro 03-789...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Krstew, E., McPherson, G. A., Malta, E., Molenaar, P., Raper, C.
Формат: Artigo
Язык:Inglês
Опубликовано: Nature Publishing Group 1984
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC1987030/
https://ncbi.nlm.nih.gov/pubmed/6145474
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