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Muscarinic activity of McN-A-343 and its value in muscarinic receptor classification.

The affinity and potency of McN-A-343 (4-(m-chlorophenyl-carbamoyloxy) -2-butynyltrimethylammonium chloride) has been assessed at a range of M1 and M2 muscarinic receptors. McN-A-343 was shown to act as a full agonist at M2 receptors present in the guinea-pig isolated taenia caeci (-log EC50 = 5.14)...

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Dettagli Bibliografici
Autori principali: Eglen, R. M., Kenny, B. A., Michel, A. D., Whiting, R. L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1987
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1917196/
https://ncbi.nlm.nih.gov/pubmed/2437988
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