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Dermorphin analogues containing D-kyotorphin: structure-antinociceptive relationships in mice.

The antinociceptive effects of synthetic dermorphin and its analogues containing D-Arg in position 2 injected into the lateral cerebroventricle were examined in conscious mice. Intracerebroventricular (i.c.v.) administration of dermorphin and [D-Arg2] dermorphin produced potent and long-lasting anti...

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Autors principals: Kisara, K., Sakurada, S., Sakurada, T., Sasaki, Y., Sato, T., Suzuki, K., Watanabe, H.
Format: Artigo
Idioma:Inglês
Publicat: 1986
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1916917/
https://ncbi.nlm.nih.gov/pubmed/2869809
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