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Effects of Piperaquine, Chloroquine, and Amodiaquine on Drug Uptake and of These in Combination with Dihydroartemisinin against Drug-Sensitive and -Resistant Plasmodium falciparum Strains

Piperaquine is being developed as a long-acting component in artemisinin combination therapies. It was highly active in vitro and drug interaction studies showed that dihydroartemisinin combinations with piperaquine, chloroquine, and amodiaquine were indifferent tending toward antagonism. Competitiv...

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Detalles Bibliográficos
Main Authors: Fivelman, Quinton L., Adagu, Ipemida S., Warhurst, David C.
Formato: Artigo
Idioma:Inglês
Publicado: American Society for Microbiology 2007
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC1891407/
https://ncbi.nlm.nih.gov/pubmed/17404003
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01479-06
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