A carregar...

The Role of Fluorine Substitution in the Structure-Activity Relationships (SAR) of Classical Cannabinoids.

A facile synthesis of 1-fluoro-1-deoxy-Δ8-THC analogs with side-chains seven carbons in length, in the alkane/ene/yne-series (6, 5 and 4), was achieved from 1-fluoro-3,5-dimethoxybenzene (1). In vitro studies show that substitution by a fluorine has a significant detrimental effect on CB1 binding wh...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Crocker, Peter J., Mahadevan, Anu, Wiley, Jenny L., Martin, Billy R., Razdan, Raj K.
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1855243/
https://ncbi.nlm.nih.gov/pubmed/17257842
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2007.01.006
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!