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Non classical, multiple-site interaction of [3H]-prazosin with the alpha 1-adrenoceptor of intact BC3H1 cells.

1. In intact BC3H1 cells the EC50 of noradrenaline (NA) for the inositol phosphate response measured at 37 degrees C (EC50 = 193 nM) was much lower than its apparent dissociation constant (Ki37 degrees C = 83.211 microM) determined at this temperature by [3H]-prazosin binding. 2. After pretreatment...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Sladeczek, F., Kirk, C. J., Bockaert, J., Schmidt, B. H.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 1989
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC1854612/
https://ncbi.nlm.nih.gov/pubmed/2551439
Etiketak: Etiketa erantsi
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