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The physiological relevance of low agonist affinity binding at opioid mu-receptors.

1. Inhibition constant (Ki) were determined for a range of opioid standards using two binding assays; [3H]-[D-Ala2, MePhe4, Gly-ol5]enkephalin ([3H]-GLYOL) binding to guinea-pig brain membranes in HEPES buffer and [3H]-naloxone binding to rat whole brain membranes in Krebs/HEPES buffer. 2. These val...

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Bibliografski detalji
Glavni autori: Carroll, J. A., Shaw, J. S., Wickenden, A. D.
Format: Artigo
Jezik:Inglês
Izdano: 1988
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1854000/
https://ncbi.nlm.nih.gov/pubmed/2840167
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