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Absolute Binding Free Energy Calculations Using Molecular Dynamics Simulations with Restraining Potentials

The absolute (standard) binding free energy of eight FK506-related ligands to FKBP12 is calculated using free energy perturbation molecular dynamics (FEP/MD) simulations with explicit solvent. A number of features are implemented to improve the accuracy and enhance the convergence of the calculation...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Wang, Jiyao, Deng, Yuqing, Roux, Benoît
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Biophysical Society 2006
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC1578458/
https://ncbi.nlm.nih.gov/pubmed/16844742
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1529/biophysj.106.084301
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