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Inhibition of heterologously expressed cystic fibrosis transmembrane conductance regulator Cl(−) channels by non-sulphonylurea hypoglycaemic agents

1. Hypoglycaemia-inducing sulphonylureas, such as glibenclamide, inhibit cystic fibrosis transmembrane conductance regulator (CFTR) Cl(−) channels. In search of modulators of CFTR, we investigated the effects of the non-sulphonylurea hypoglycaemic agents meglitinide, repaglinide, and mitiglinide (KA...

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Detalhes bibliográficos
Main Authors: Cai, Z, Lansdell, K A, Sheppard, D N
Formato: Artigo
Idioma:Inglês
Publicado em: 1999
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1571594/
https://ncbi.nlm.nih.gov/pubmed/10498841
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702748
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