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The putative melatonin receptor antagonist GR128107 is a partial agonist on Xenopus laevis melanophores
1. GR128107 (3-(1-acetyl-3-methyl-piperidine)-5-methoxyindole) has previously been reported to be a competitive melatonin receptor antagonist in blocking melatonin inhibition of [(3)H]-dopamine release from rabbit retina, a response mediated by the MT(2) receptor subtype. 2. GR128107, like melatonin...
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| Hlavní autoři: | , |
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| Médium: | Artigo |
| Jazyk: | Inglês |
| Vydáno: |
1999
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| Témata: | |
| On-line přístup: | https://ncbi.nlm.nih.gov/pmc/articles/PMC1565880/ https://ncbi.nlm.nih.gov/pubmed/10205014 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702404 |
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