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The putative melatonin receptor antagonist GR128107 is a partial agonist on Xenopus laevis melanophores

1. GR128107 (3-(1-acetyl-3-methyl-piperidine)-5-methoxyindole) has previously been reported to be a competitive melatonin receptor antagonist in blocking melatonin inhibition of [(3)H]-dopamine release from rabbit retina, a response mediated by the MT(2) receptor subtype. 2. GR128107, like melatonin...

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Bibliografski detalji
Glavni autori: Teh, Muy-Teck, Sugden, David
Format: Artigo
Jezik:Inglês
Izdano: 1999
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1565880/
https://ncbi.nlm.nih.gov/pubmed/10205014
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702404
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