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Pharmacological analysis of G-protein activation mediated by guinea-pig recombinant 5-HT(1B) receptors in C6-glial cells: similarities with the human 5-HT(1B) receptor

1. The guinea-pig recombinant 5-hydroxytryptamine(1B) (gp 5-HT(1B)) receptor stably transfected in rat C6-glial cells was characterized by monitoring G-protein activation in a membrane preparation with agonist-stimulated [(35)S]-GTPγS binding. The intrinsic activity of 5-HT receptor ligands was comp...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Pauwels, Petrus J, Wurch, Thierry, Palmier, Christiane, Colpaert, Francis C
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: Nature Publishing Group 1998
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC1565141/
https://ncbi.nlm.nih.gov/pubmed/9484854
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0701584
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