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Inhibition of [(3)H]-U69593 binding and the cardiac effects of U50,488H by calcium channel blockers in the rat heart

1. The calcium channel blockers (CCBs), nifedipine, nicardipine, diltiazem and verapamil, were used to displace the binding of [(3)H]-U69593 ((5a,7a,8b)-(+)-N-methyl-N-(7-[1-pyrrolidinyl]-1-oxaspiro[4,5]dec-8-yl)-benzeneacetamide), a specific κ-opioid agonist, in the rat cardiac sarcolemma. The CCBs...

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Detalhes bibliográficos
Main Authors: Zhang, Wei-Min, Wang, Hong-Xin, Xia, Qiang, Wong, Tak-Ming
Formato: Artigo
Idioma:Inglês
Publicado em: 1997
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1564545/
https://ncbi.nlm.nih.gov/pubmed/9138688
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0700985
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