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Local anesthetics. Effect of pH on use-dependent block of sodium channels in frog muscle.

Sodium currents were studied under voltage clamp in the presence of neutral, amine, and quaternary local anesthetic compounds. Use-dependent block was observed as a cumulative depression of INa seen with repetitive depolarizing test pulses applied at frequencies of 2-10s-1. With quaternary QX-314, t...

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Библиографические подробности
Главные авторы: Schwarz, W, Palade, P T, Hille, B
Формат: Artigo
Язык:Inglês
Опубликовано: 1977
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC1473363/
https://ncbi.nlm.nih.gov/pubmed/21711
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