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A new class of inhibitors of 2-arachidonoylglycerol hydrolysis and invasion of prostate cancer cells

Endogenous 2-arachidonoylglycerol (2-AG) inhibits invasion of androgen-independent prostate cancer cells. Blocking cellular hydrolysis of 2-AG to increase its endogenous concentration results in a decrease in cell invasion. A series of compounds containing a trifluoromethyl ketone (TFK) moiety or th...

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Bibliografiske detaljer
Main Authors: Nithipatikom, Kasem, Endsley, Michael P., Isbell, Marilyn A., Wheelock, Craig E., Hammock, Bruce D., Campbell, William B.
Format: Artigo
Sprog:Inglês
Udgivet: 2005
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC1450257/
https://ncbi.nlm.nih.gov/pubmed/15919052
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbrc.2005.05.049
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