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Spectroscopic analyses of the binding kinetics of 15d-PGJ(2) to the PPARγ ligand-binding domain by multi-wavelength global fitting
PPARγ (peroxisome proliferator-activated receptor γ) is a nuclear receptor that is activated by natural lipid metabolites, including 15d-PGJ(2) (15-deoxy-Δ(12,14)-prostaglandin J(2)). We previously reported that several oxidized lipid metabolites covalently bind to PPARγ through a Michael-addition t...
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| Autors principals: | , , , , |
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| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
Portland Press Ltd.
2006
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC1360728/ https://ncbi.nlm.nih.gov/pubmed/16236024 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20050930 |
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